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AASraw inopa marudzi ehuremu hwekurasikirwa nehupfu nehupfumi hwakagadzikana, zvose zvinogadzirwa zvinopedzwa pasi peCGMP mutemo uye hutano hunogona kuteverwa chero nguva. Mukuwedzera, iyo yakawanda yekuraira inogona kutsigirwa nemutengo unokwikwidza.

Orlistat Inoshanda Sei Seweya Wekurasikirwa Zvinodhaka

Tenga Weight Loss Powder

1.Weight Loss Drug History

Yokutanga kurasikirwa kwemishonga, iyo inonzi mafuta ekuchera panguva iyoyo, yakasvika pakupedzisira kwe1800s. Kunyange zvazvo mishonga iyi yakakonzera mamwe madhara akaipa, yakaramba ichiwanikwa kuti ishandiswe kusvikira ku1960s.

Mishonga mitsva inozivikanwa seDinroprophenol yakaiswa muZ1930 uye yakava yakakurumbira pakugadzirisa kurasikirwa. Iyo mishonga yakabudisa hutemogenic mukati momuviri, kuita kuti kurasikirwa kuwedzere.

Pakati pe-1950s, amphetamine yakavapo uye yakashanduka kuve kurasikirwa nemishonga yekusarudza. Yakaita kuti kurasikirwa kwemahombekombe kuve kukanganisa nekudzivisa kudya. Zvinosuruvarisa, yakawedzera ngozi yepemmonia yeupempersion, zvichiita kuti ibve kubva pamusika mu1968.

Mune 1970s, ephedrine yakave yakarongerwa kurapwa kwekurema. Mishonga iyi, zvisinei, yakakonzera kushushikana kwakashata kwakazoita kuti iziviswa kuti inotyisa.

Muna 1973, fenfluramine yakagamuchirwa sekuti kurasikirwa kwekureruka kuwedzera. Kuzivikanwa kwaro kwakasimudzirwa mu1992 apo yaisanganiswa ne phentermine kuumba kurasikirwa kwemazizi kunonzi fen-phen. Zvinosuruvarisa kuti mishonga iyi yakakonzera zvimwe zvinetso zvakashata, izvo zvakaita kuti zvibve pamusika mu1997. Muzana remakore reC21, kurasikirwa kwechiremera chemishonga, zvakawanda zvakabva pamaruva emiti, yakazara mumusika.

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Yakavimbika Tsime

PubMed Central

Inoremekedzwa dhatabhesi kubva kuNational Institutes of Health
Enda kunzvimbo

2.Weight Loss Drug Classification

Kurema kwekurasikirwa zvinodhaka zvinongororwa kuva zvikamu zvitatu zvakakura maererano nemaitiro avo ekuita uye zvinotevera:

 

(1) Appetite suppressant (Zvokudya)

Zvinodhaka zvinoderedza kudya zvokudya zvinonzi sympathomimetic agents. Vanowanzodzvinyirira chido apo vachiita kuti satiety isati yasvika. Satiety ndiyo "yakazara" kunzwa kana kugutsikana kunowanikwa pakutora zvokudya. Maitiro ekudzvinyirira anoshanda nekutevedzera neurotransmitter muhuropi hwemunhu inodzora chido, inozivikanwa sa noradrenaline (NA).

 

Iyi mishonga inogovera chimiro chemakemikari yakafanana ne NA uye inogona; semugumisiro sunga kune imwechete receptors se noradrenaline. Iyo mishonga inovandudzawo noradrenaline basa mu "feeding centre" yehuropi hwevanhu, hypothalamus. Iyo hypothalamus yemunhu inodzora chiyero chesimba muhurongwa hwemuviri. Iwo ruzivo nezve ega ega emagetsi ezvitoro anogadzirwa mu hypothalamus iyo inodzora kudya kwekudya uye kuda kudya. Noradrenaline kusunga uye kuita mu hypothalamus kune kuderedza mhedzisiro pakuda kudya. Mishonga yakadai inosanganisira:

❶ Lorcaserin HCL(Belviq) CAS: 1431697-94-7

❷ Rimonabant HCL CAS: 158681-13-1

❸ DNP CAS: 119-26-6

 

(2) Fat Burning

Mafuta anopisa uremu zvinodhaka zvinogona kubatsira kurasikirwa kwemafuta nekuderedza zvishuwo, kuwedzera metabolism, uye kuchengetedza kudya kune hutano. Ivo vanogona zvakare kukwirisa kugona kwekurovedza muviri nekuwedzera simba uye kutarisa. Mishonga yakadai inosanganisira:

❶ Synephrine CAS: 94-07-5

❷ DMAA/1,3-Dimethylpentylamine CAS: 13803-74-2

 

(3) Kuvandudza kudya

Izvi zvinorema kurasikirwa nemishonga zvinoshanda nekupindira nekwanisi yekugadzirisa chirongwa ichi kuti iwane zvimwe zvokudya muzvokudya. Somuenzaniso, Orlistat inozivikanwa kuvhiringidza kuparara kwemafuta uye naizvozvo inodzivisa kudya kwemafuta. Zvimwe zvidimbu zvakawanda zvakashandiswa mukuderedza caloric absorption uye kudzivisa kudya. Muchikamu ichi, tichakurukura zvakawanda pamusoro pemishonga yakadaro inotevera:

❶ Orlistat CAS: 96829-58-2

❷ Cetilistat CAS: 282526-98-1

Kurasika Kwemafuta upfu peji mufananidzo01

3.Iyo 3 Inonyanya Kuzivikanwa Weight Loss Poda Mumusika

(1) Orlistat CAS: 96829-58-2

Orlistat inonyanyisa pancreatic uye gastric lipase inhibitor. Zvose zvekudya zvinonzi triglycerides zvinogadziriswa nemubatsiro we pancreatic uye gastric lipases. Iyo inopisa enzymatically inoputsa pasi triglycerides muhusununguko husina mafuta acids iyo inogona kuve yakabatwa mumatumbo maduku. Gastric uye pancreatic lipase inhibitors zvakagadzikana nesangano repancreatic uye gastric lipases mu lumen yemukati muduku uye mudumbu zvichiita kuti ma enzymes aregone kushanda zvakanaka.

Kuburikidza nekudzivisa kwechiito chezviputika izvi, kudya kwemafuta kunodya kunodzivirirwawo, uye triglycerides inowedzerwa mumucheka. Orlistat kurasikirwa nemishonga kunodzivirira kumativi ose 30 muzana yemafuta ane utano kubva pakudya kubva pakupinda mumuviri wemunhu (apo 30 muzana yezvokudya muzvokudya zvinopiwa ne triglycerides). Ivhareji inorema kuderedza mushure megore rimwe nekubatanidzwa kweXenical (orlistat) uye kuchinja mumararamiro ehupenyu kune kambani 8.5 kg.

Pamwe nekudzikisa kudyidzana kwezvokudya zvinonzi triglycerides, orlistat kurasikirwa kwehupfu kwakawanikwa ku:

  • Iva nemigumisiro yakanaka pahutano hweropa;
  • Deredza kunyura kwecholesterol uye saka cholesterol mazinga (pamwe chete neLDL cholesterol);
  • kuwedzera insulini kuramba; uye
  • Wedzera glycemic control.

Inofungidzirwa zvakanyanya kuti orlistat's gastrointestinal adverse effects inoita nenzira yakafanana nekusimbisa kwakashata, iyo inokurudzira avo vari pamushonga uyu kuti vatevedzere zvakasimba kune kudya kwemafuta mashoma.

 

(2) Cetilistat CAS: 282526-98-1

Cetilistat inoshandiswa nemuromo, inoveli, pancreatic uye gastrointestinal lipase inhibitor. Cetilistat uremu kurasikirwa mushonga mushonga unogadzirwa kurapa kufutisa. Inoshanda nenzira yakafanana semushonga wakambokurukurwa kare unozivikanwa seXenical (orlistat) nekudzora pancreatic lipase, iyo enzyme inoputsa triglycerides mumatumbo edu. Pasina aya ma enzymes, triglycerides kubva muchikafu chedu inodzivirirwa kubva pakugayiwa mumahara emafuta acids anogona kutorwa uye anobviswa kubva mumuviri usina kugezwa.

Mumakiriniki ekuedzwa kunosanganisira varwere vanorema vasina chirwere cheshuga 2 uye mune varwere vakanyanya vanorarama nechirwere cheshuga 2. Apo Cetilistat kurasikirwa kwemafuta kwakapiwa kwemavhiki gumi nemaviri, zvakakosha zvikuru kuderedza muviri, huwandu hwecholesterol, serum low-density lipoprotein cholesterol nokukurumidza pakuenzanisa ne placebo.

Izvo zviyero zvevarwere vanorema zvakaratidza kuderedzwa kukuru muhutano hwekutanga hwemuviri wehutori huwandu hwe5 hwepamusoro hwakanga hwapamusoro pane zvese zvakashanda zvichienzaniswa ne placebo. Mukuwedzera kwehuwandu hwevanhu vane chirwere cheshuga, HbA1c (glycosylated hemoglobin) mazinga akanyanyawo kuderedzwa. Cetilistat kuora kurasikirwa kwemishonga kwakaratidza kuenzanisa kusvika kune zvinorwadza zvakanyanya, zvinowanzokonzera steatorrhea (kushaya muviri) uye ine chirwere chakanyanya kupfuura icho chiri mu orlistat. Iyi mishonga yakanga ichangobva kugamuchirwa muJapan kunobata kuneta nekumwe matambudziko.

 

(3) Lorcaserin HCL(Belviq) CAS: 1431697-94-7

Lorcaserin HCl zvinodhaka zvinodhaka kudzora metabolism uye chido. Mushonga uyu wakabvumidzwa neFDA mugore ra2012 kune vanhu vane BMI inopfuura makumi matatu, uye kune varwere vane Body Mass Index yemakumi maviri nenomwe kana kupfuura vanewo high cholesterol, blood pressure, uye Type 30 chirwere cheshuga. Mushonga unoshandawo kusimudzira serotonin 27CV receptor muuropi hwemunhu iyo inogona kubatsira varwere kuti vanzwe vakaguta mushure mekutora zvishoma. Mune miedzo yezvokurapa, 2% yevanhu vakuru (pasina rudzi rwechipiri chirwere cheshuga) vakarasikirwa nepamusoro pe2% yehuremu hwemuviri wavo, mukuenzanisa ne38% yevanhu vakuru vanobatwa ne placebo. Sezvo sibutramine powder yakarambidzwa muChina, lorcaserin hcl powder ndiyo inonyanya kushandiswa mumusika uye vatengesi vakawanda vakazvipira pakugadzirwa kwemishonga yekurasikirwa vanosarudza kushandisa lorcaserin hcl powder.

( 8 17 3 )↗

Yakavimbika Tsime

PubMed Central

Inoremekedzwa dhatabhesi kubva kuNational Institutes of Health
Enda kunzvimbo
Kurasika Kwemafuta upfu peji mufananidzo02

4.How To Kutenga Inobudirira Weight Loss Powder Online?

Sezviri kuonekwa kubva pane zvatakanyatsokurukurirana, pane zvakawanda zvinorema kurasikirwa nemishonga kunze uko izvo zvakabva kune dzakawanda zvakasiyana-siyana masangano. Mishonga yemishonga iyi yakawanikwa ichibudirira, uye dzimwe dzadzo dzakagamuchirwa nemitemo dzakasiyana-siyana dzakadai seDefA neJapane, kutaura zvishomanana, pakurapa kuneta.

Mushure mekupedza maawa akawanda tichitsvaga zvinodhaka zvekuderedza uremu, takakwanisa kuona mashoma 2018 World's Best-Selling Weight Loss Powder Supplements. Izvi zvinorema kurasikirwa poda zvinowedzera zvinosanganisira orlistat uremu kurasikirwa poda uye lorcaserin uremu kurasikirwa poda. Kusiyana nehuremu hwehuremu hwekuwedzera hunowanikwa pane chero chitoro chemishonga, iyi mishonga yekurasikirwa nehuremu yakatemwa nenyanzvi dzekurapa yapfuura makore ekuyedzwa kuti vawane chitambi chekubvumidzwa kubva kuFDA nedzimwe nzvimbo dzakati wandei. Isu tinokurudzira zvikuru kuti uedze mishonga iyi nekuti yakaratidza kuti haina kungoshanda chete asiwo yakachengeteka kushandisa.

Iwe unogona kubvunza kuti ungatenga sei uremu hunorema hupfu orlistat powder uye lorcaserin hcl powder. Kune akawanda ekurasikirwa nehuremu vatengesi pamhepo uye vanoda kufunga kuti ndeipi yakakunakira iwe. Iwe unofanirwa kubhadhara zvakanyanya kumhando yezvigadzirwa uye kuti zvinogona kutumirwa kwauri zvakachengeteka, kana iwe uchida kutenga uremu kurasikirwa hupfu muhuwandu, iwe unofanirwa kuziva kana yavo yekugovera system uye kana yakagadzikana, funga nezve kutora sampuli odha isati yawanda. odha, tora kuti uedze kunyanzvi 3rd-Labs uye tarisa kunaka. Zvakadaro, kuwana mhando yepamusoro mupi hazvisi zvinhu zviri nyore, iwe unofanirwa kuisa yakawanda nguva nesimba pazviri.

Kutenga genius uremu kurasikirwa / kudya mushonga mbishi poda inoda kungwarira zvakanyanya, kunyanya nekutenga online online. Kune maviri akawanda masosi anoti anopa zvinhu zvehungwaru asi anoratidzwa sema scammers. AASraw inopa uye inopa chete genius zvinhu. Iyo inozivikanwa nevakawanda vevanhu nemakambani, vanogona kupa huwandu hwekuremerwa hupfu hupfu, hwakadai sa lorcaserin hcl, orlistat, Cetilistat. Iyo nyanzvi yekuyedza mishumo inogona kugoverwa uye inoratidza 98% maminetsi kuchena. Unogona kutaura neaasraw sales kuti uwane mamwe mashoko online!

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Yakavimbika Tsime

PubMed Central

Inoremekedzwa dhatabhesi kubva kuNational Institutes of Health
Enda kunzvimbo

FAQ

1.Lorcaserin inobatsira sei kuti uremerwe uremu?

Kuti uremerwe uremu, Lorcaserin inoshanda nekukanganisa manzwiro emuviri ekunzwa akazara nekuchinja serotonin mazinga muuropi. Ndiyo nzira iyo Lorcaserin inogona kushanda kurapa kupindwa muropa neopioid.

2.Is lorcaserin hcl powder inodzorwa here?

Kunyange zvazvo isiri iyo inokurudzira, lorcaserin inogona kukonzera kuderedzwa kwezvinodhaka uye kushatiswa. Nokuda kwechikonzero ichi, Drug Enforcement Administration (DEA) yakarongedza iri pasi peMutemo weDzimwe Chetsika paHatendi IV.

 

Saka, vanogadzirisa sei miyero yako? Ndichatsanangura. Kunyanya kudarika kunogona kunge kwakangoerekana kwaitika asi zvinogona kunge zvakare kushandiswa kwechinangwa chokukurudzira mushandisi. Kuti uwane hutano, iwe unogona chete kugadzirisa zvinyorwa zvezviverengero zvishoma.

Mimwe yemigumisiro ye lorcaserin inosanganisa maitiro, kunzwa 'kukwirira', kudengenyeka, kana kufara. Muzviitiko zvishomanana, vamwe varwere vakasiya chirwere ichi vakaratidza zvimwe zviratidzo zvekudzoka. Zvose izvi zvinokwana uchapupu hwokuti mishonga inogona kukonzera kushungurudza kwepfungwa.

3.Is uremu-kurasikirwa nemishonga lorcaserin hcl yakachengeteka?

Chidzidzo chikuru chakawana migumisiro inovimbisa yekuchengetedzwa kwemishonga inorema-kurasikirwa inowanika muUnited States.Chidzidzo, chakabudiswa muNew England Journal of Medicine, inoti vanhu vakuru vachishandisa mushonga lorcaserin vakarasikirwa nehuwandu hwe4kg (8.8lb) pamusoro pe40 mwedzi. Inoti mushonga uyu, unoshanda nekudzvanyirira kudya, hauise vanhu panjodzi huru yekunetsekana nemoyo. Asi nyanzvi dzinosimbisa kukosha kwekuchinja kwehupenyu hwenguva refu pakuwana uremu hunobudirira.Lorcaserin yave iripo muUnited States kwemakore akawanda pasi pezita rokuti Belviq, asi haisati yabvumirwa kushandiswa muEurope.

4.Is Orlistat inoshanda pakurasikirwa uremu?

Orlistat inoshanda nekudzivirira mafuta kubva muchikafu chaunodya kubva pakupinzwa mumuviri wako. Mafuta aya anozobuda mumuviri kuburikidza netsvina yako.

Kuti Orlistat ishande, inofanira kushandiswa pamwe chete nemamwe maitiro ekuderedza uremu. Izvi zvinosanganisira chirongwa chekurovedza muviri nguva dzose uye chirongwa chekudya chine utano. Kana yakatorwa pachayo, Orlistat inogona kusaderedza uremu, sezvo isingapise mafuta aripo.Kana yakashandiswa pamwe chete nemamwe maitiro ekuderedza uremu, Orlistat yakaratidza kuti inoshanda pakubatsira uremu.

Imwe ongororo yakawana kuti vanhu vakatora Orlistat uye vakachengeta kudya kwakaderera-koriori vakarasikirwa neavhareji 1.25 dombo (8.1kg) pagore, iyo yaive 6lb (2.8kg) kupfuura avo vasina kutora Orlistat panguva imwecheteyo. Imwe ongororo yakawana kuti 743 varwere vakafuta vanotora Orlistat yekurasikirwa nehuremu vaive varasikirwa neavhareji 10.3kg yehuremu mushure megore rimwe. Izvi zvakasiyana nevarwere ve6.1kg vasingatore Orlistat vakarasika.

Zvimwe zvidzidzo zvakaonawo kuti vanhu vanotevera nzira yekurapa iyi vanogona kurasikirwa nechikamu chegumi kubva muzana chehuremu hwemuviri wavo mugore.

5.Ndiani anofanira kushandisa orlistat powder?

Orlistat yekurasikirwa kwehuremu inonyanya kutorwa nevaya vanonetseka kuderedza uremu kuburikidza nedzimwe nzira. Usati watanga Orlistat, unofanira kutanga waedza kuderedza uremu kuburikidza nekoriori-inodzorwa nekudya uye kurovedza muviri nguva dzose. Iwe unofanirwawo kufunga nezvekurega kusvuta uye kuderedza kunwa kwako doro usati watora mushonga. Mushure mekutora Orlistat kwemavhiki mashoma, unogona kutarisira kuona kurasikirwa kukuru kwehuremu. Mari chaiyo inosiyana pakati pevanhu, zvichienderana nekudya kwavo uye maitiro ekurovedza muviri.

6.Orlistat powder wongororo: pamberi uye shure

Zak (4th, Kurume. 2021): Ichi ndicho chirongwa chekutanga chekurasikirwa kwehuremu chandakakwanisa kunamatira. Ndinokurudzira zvikuru Orlistat powder. Kana iwe usingade "maitiro ekurapa", saka iwe unonyatso tarisa mafuta ako ekudya! Handikwanise kutaura zvakakwana nezveOrlistat poda. Ndakaona kuti ndinogona kuva nezvokudya zvakasiyana-siyana - asi chikamu chikuru ndicho kiyi!

 

Jimmy(16 Kubvumbi 2020): Mavhiki e3 kusvika zvino akanaka kubva pandinotenga orlistat poda online uye edza zvimwe. Ndiri kuonda zvishoma nezvishoma zvinova zvandinoda kuti ndisaite yoyo affect. RAMBA pakudya kwako kwakaderera kwemafuta. Ndakadya pizza rimwe zuva ndokutevera nezvimedu zviviri zvemangwanani uye ndakabuda mafuta eorange paibuda gasi kana panguva yekufamba. Hongu zvinokuzivisa iwe kana wadya zvakanyanya kana zvisiri izvo. Verenga macalories ako idya miriwo yakawanda uye michero. Inwa mvura. After reading others side affects zvinondibatsira kunamatira Alli nekuti pazvinoitika unokwenya musoro uchiti UhUh, oh no, you laughing me.

 

Bob(24 Sep. 2021): Ndinorasikirwa nemakirogiramu matanhatu muvhiki imwe ne orlistat powder .. asi ndinodya zvokudya zvine utano mon thru fri: zvokudya zvakaderera mafuta uye zvishoma makorikori uye vhiki yevhiki ndinodya chero chinhu chine mwero. Zvakare, ini ndinofamba 6 maminetsi mazuva ese uye ndinotamba tennis maawa matatu ndakagara.

Sekupupura kuri pamusoro apa, zviitiko zvevatengi vedu zveOrlistat sekurapa-kuderedza uremu zvakanaka zvakanyanya. Heano mashoma eakakosha maitiro evatengi vedu ongororo yeOrlistat yakasimbiswa:

♦ Inoshanda pakubatsira varwere kuderedza uremu

♦ Yakanakira kutangisa uremu chirongwa

♦ Inobatsira pakuderedza uremu zvishoma nezvishoma asi zvakatsiga pavhiki

♦ Zvinobatsirawo kuderedza cholesterol

Pakazara, vatengi vedu vanonongedza kuOrlistat senzira yakavimbika uye inoshanda yekuderedza uremu.

7.Ndeipi mhedzisiro yeorlistat?

Zvinowanzoitika mhedzisiro yeOrlistat

Iwo akajairika mhedzisiro yeOrlistat anowanzo kukanganisa akatenderedza munhu mugumi vanhu. Izvi zvinosanganisira zviri pazasi, asi zvinonyanya kuitika kutemwa nemusoro:

▪ Tsvina ine mafuta kana yakakora kana zvinobuda zvine mafuta kubva kuburi rako — tarisa mavara ane mafuta pachipfeko chako chemukati.

▪ Kubuda ura nokukurumidza

▪ Kuwedzera flatulence, dzimwe nguva nekubuda

▪ Kutemwa nemusoro

▪ Zvirwere zvepamusoro (RTIs), zvakadai sedzihwa

▪ Kurwadziwa nemudumbu kana kusagadzikana

Zvese izvi mhedzisiro ndezvenguva pfupi uye zvinofanirwa kupfuura nekufamba kwenguva. Zvisinei, kana ukasangana navo kwenguva yakareba, kana kuti vanowedzera kuipa, bvunza chiremba wako pakarepo.

 

Zvishoma zvakajairika mhedzisiro yeOrlistat

Migumisiro yeOrlistat pazasi haina kunyanya kuwanda pane idzo dzakanyorwa pamusoro uye dzinosanganisira:

▪ Tsvina yakapfava

▪ Kusazvidzora kwetsvina

▪ Kusagadzikana kwemazino

▪ Kuzvimba — izvi zvinowanzoitika kuvanhu vane chirwere cheshuga cherudzi rwechipiri

▪ Kusatevera nguva

▪ Kuneta

▪ Zvirwere zvepasi pekufema

▪ Marwadzo kana kuti kusanzwa zvakanaka

Kana iwe ukasangana nechero yeiyi mhedzisiro kwenguva yakareba kana kuti zviratidzo zvako zvinotanga kuipa, taura nachiremba wako nekukurumidza sezvinobvira.

8.Ndingaderedza sei migumisiro yeOrlistat?

Mazhinji mhedzisiro yeOrlistat ndeyenguva pfupi uye inoenda nenguva. Kana mhedzisiro yako isingaendi, taura nachiremba wako nekukurumidza sezvinobvira. Zvinokwanisika kuderedza migumisiro yeOrlistat nekuyera kuti unodya mafuta akawanda sei mukudya kwega kwega.

Orlistat inoshanda nekumisa mafuta muchikafu chako kubva pakunyudzwa mudumbu. Inodzinga chero mafuta asina kunyura kuburikidza nemuura. Zvisinei, Orlistat inogona chete kubvisa mafuta akawanda pakudya. Nekuda kweizvozvo, kana iwe ukadya chikafu chine anopfuura 1-15 magiramu emafuta, unogona kusangana neOrlistat's side effects kakawanda. Kuti uderedze mhedzisiro yeOrlistat, usadya inopfuura 1-15 magiramu emafuta pakudya kana uri kutora Orlistat 120 mg capsules.

Iwe unogona zvakare kuderedza mhedzisiro yeOrlistat nekunamatira kune chaiyo dosage yeOrlistat. Kutora kupfuura yakakurudzirwa dosage yeOrlistat mushure mekudya kunowedzera mhedzisiro yayo, saka namatira kune dosi inokurudzirwa.

9.How kushandisa Kotilistat powder kurapa kuneta?

Kuwedzera kwekuwedzera kwekuneta kwakakonzera kutsvaga kwemishonga yekurapa chirwere ichi. Nzira dzakasiyana-siyana dzokurapa dzave dzichiongororwa, kusanganisira:

▪ Serotonin uye noradrenaline reuptake inhibitors (anorectic agents)

▪ Lipase inhibitors

▪ b 3-adrenoreceptor agonists

▪ Leptin agonists

▪ Melanocortin-3 agonists

▪ Endocannabinoid receptor antagonists

 

Cetilistat powder inonzi lipase inhibitor, ine maitiro akafanana ekuita kuRoche's anti-obesity mishonga orlistat powder yakagamuchira mvumo yekutonga mu 1997. Mishonga iyi inoshanda mumakumbo emimba kuti inhibit lipases, ma enzymes anobatanidzwa mukuparara kwemafuta ekudya. Nekudzivisa kuparara uye kunotevera kunyura kwemafuta kubva mumatumbo, lipase inhibitors inoderedza kudya kwemafuta uye macalorie, nokudaro kubatsira kurasikirwa kwemafuta.

10.Orlistat Powder Vs Cetilistat powder

Items Orlistat Upfu Cetilistat powder
CAS nhamba 96829-58-2  282526-98-1
Mechanism of action Orlistat haishande nekudzvinyirira kudya; inoderedza kuwanda kwemafuta ayo muviri wako unotora kubva kune chikafu chaunodya. Cetilistat inonzi gastrointestinal lipase inhibitor inovhara kudyiwa kwemafuta uye kunwa, zvichiita kuti kuderedza simba rekudya, uye nokudaro kuderedza uremu.
Dosage 120 mg nemuromo katatu pazuva nekudya kukuru kwega kwega kune mafuta. 120 mg katatu pazuva pakarepo mushure mekudya kwega kwega.
Zvikanganiso ▪ Gasi rinopfuura, dzimwe nguva rine mavara ane mafuta

▪ Zvitsvina zvisina kusimba, tsvina ine mafuta, kana manyoka

▪ Kugara uine tsvina kana kuti kubuda ura zvakaoma kudzora

▪ Kuzvimbirwa

▪ Kurwadziwa mudumbu

▪ Kuzvimba

▪ Zvine mafuta

▪ Zvituru zvisina kusimba

▪ Fecal incontinence

▪ Kuzvimba

▪ Marwadzo Mudumbu

▪ Zvituru zvakapfava

▪ Muromo Wakaoma

 

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Reference

[1] "FDA Nyaya Dzakazara Mhinduro Tsamba yeLorcaserin Mutsva Wemushonga Wekushandisa". 23 Gumiguru 2010. Yakachengetwa kubva kune yekutanga musi wa24 Gumiguru 2010.

[2] Higham, George (5 Chikumi 2020). "ᐅ Orlistat & Xenical: Ko Mapiritsi ekuderedza uremu Anoshanda? | e-Surgery”. e-surgery. Yakadzorerwa 9 June 2020.

[3] "Fake Alli kudya mapiritsi anogona kuunza njodzi kune hutano". CNN. 23 Ndira 2010. Yakadzorerwa 24 Ndira 2010.

[4] Yamada Y, Kato T, Ogino H, Ashina S, Kato K: Cetilistat (ATL-962), inoveli pancreatic lipase inhibitor, inosimbisa kuwedzera kwemuviri uye inovandudza lipid profiles mumakonzo. Horm Metab Res. 2008 Aug;40(8):539-43. doi: 10.1055/s-2008-1076699. Epub 2008 Chivabvu 21.

[5] Devarajan, Uma (1 Kurume 2009). "Nyaya dzemafuta". Iyo Deccan Chronicle. Yakadzorerwa 26 Mbudzi 2009.

[6] Yakashongedzwa nemavara madiki a pakurongedzerwa, uye bhaa pamusoro pei (kureva, "alī"), asi yakatorwa mazita echinyakare muchinyorwa.

[7] Pollack A (16 Gunyana 2010). "FDA Panel Inoramba Diet Pill". Iyo New York Times. Yakachengetwa kubva kune yekutanga musi wa 17 Chikunguru 2011.

[8] "Lorcaserin Shandisa Panguva Yepamuviri". Drugs.com. 4 Mbudzi 2019. Yakadzorerwa 14 Ndira 2020.

[9] Padwal, R (2008). "Cetilistat, itsva lipase inhibitor yekurapa kuneta". Ikozvino Maonero muKuongorora Zvinodhaka. 9 (4): 414–21. PMID 18393108.

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