Lorcaserin HCL upfu Mugadziri & Factory
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Lorcaserin HCL powder

Rating: SKU: 1431697-94-7. Category:

AASraw inyanzvi inogadzira Lorcaserin hydrochloride poda yakasvibirira ine labhu yakazvimiririra uye fekitori hombe serutsigiro, zvese zvinogadzirwa zvichaitwa pasi peCGMP mutemo uye trackable quality control system. Iyo yekugovera sisitimu yakagadzikana, zvese zvekutengesa uye zvekutengesa maodha zvinogamuchirwa.Welcome to order from AASraw!

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Product Description

Lorcaserin hydrochloride Powder Vhidhiyo-AASraw

 


Raw Lorcaserin hydrochloride Powder Basic Characters

Name: Lorcaserin hydrochloride powder
CAS: 1431697-94-7
Molecular Formula: C11H15Cl2N
Molecular Kurema: 232.1525
Melt Point: 212 ° C
Storage Temp: -20 ℃
Color: White powder

 


chii is Lorcaserin hydrochloride Powder?

Lorcaserin hydrochloride inonzi hydrochloride inowanikwa nekuita kwe lorcaserin ine imwe yakaenzana nehydrochloric acid. Inoshandiswa semushonga unorwisa kufutisa. Iine basa se serotonergic agonist uye chido chekuora mwoyo.

Lorcaserin hydrochloride powder inokanganisa zviratidzo zvemakemikari muuropi iyo inodzora kudya. Lorcaserin HCL powder inoshanda nekukubatsira kuti unzwe wakakwana nezvokudya zviduku.Lorcaserin hydrochloride powder inoshandiswa pamwe chete nekudya uye kurovedza muviri kurapa kuneta.Lorcaserin hydrochloride powder dzimwe nguva inoshandiswa kurapa kuneta kunogona kunge kwakabatana nechirwere cheshuga, high cholesterol, kana kuwedzerwa kweropa. .

Chii chinonzi Lorcaserin hydrochloride yakanaka?

Lorcaserin hydrochloride inoshandiswa kubatsira vanhu vakuru vane uremu kana kuti vane uremu uye vane matambudziko ehutano ane uremu kuti vaderedze uremu uye varambe vachidzosa uremu ihwohwo. Lorcaserin inofanira kushandiswa pamwe chete nekuderedza calorie kudya uye chirongwa chekurovedza muviri. Lorcaserin iri mukirasi yemishonga inonzi serotonin receptor agonists. Inoshanda nekuwedzera manzwiro ekuzara kuitira kuti zvokudya zvishoma zvidyiwe.

Lorcaserin hydrochloride inoshandiswa pamwe chete nekuderedzwa-koriori kudya uye kurovedza muviri kwakakodzera kukubatsira kuti uremerwe uremu. Inoshandiswawo kune vanhu vakafuta vanogonawo kuva nechirwere cheshuga, high blood pressure, high cholesterol, kana chirwere chemwoyo.

The Benefits yeLorcaserin hydrochloride

Lorcaserin hydrochloride mushonga unoitwa nemuromo unokurudzira kuora muviri. Inoshandiswa nekudya uye kurovedza muviri muvanhu vakuru vanorema vane dambudziko rehutano rine chekuita nehuremu kana vanhu vakuru vakafutisa kuti vadzike uremu uye vazvichengetedze.

Lorcaserin hydrochloride inonzi serotonin 2C (5-HT2C) inogamuchira agonist. lorcaserin inofungidzirwa kuti inosarudza kukurudzira 5-HT2C receptors mu hypothalamus, nzvimbo yeuropi inozivikanwa kuti inobata basa guru mukugadzirisa nzara uye kudya kwekudya. Nokuita izvi zvinogamuchirwa, lorcaserin inogona kuderedza kushandiswa kwezvokudya nekuderedza kudya uye kuita kuti munhu anzwe akaguta kunyange mushure mekudya zvokudya zvishoma kudarika nguva dzose.

Lorcaserin hydrochloride inonzi serotonin 2C receptor agonist inoratidzwa nokuda kwekurapa kwehutano husingagumi kune vanhu vakuru vane body mass index (BMI) ye30 kana yakakura (yakanyanya) sekuwedzera kune yakaderedzwa-calorie kudya uye kurovedza muviri. lorcaserin inobvumirwawo kuti ishandiswe nevanhu vakuru vane BMI ye27 kana yakakura (yakawandisa) uye vane imwe yehutano hunoenderana nehuremu hwakadai sehupamhi hweropa (hypertension), rudzi rwe 2 chirwere cheshuga, kana high cholesterol (dyslipidemia).

Lorcaserin hydrochloride inoshandiswa semushonga unorwisa kufutisa

Kufutisa chinhu chakakosha pahutano chinoda nzira dzakachengeteka uye dzinoshanda dzekugadzirisa denda rekufutisa. Lorcaserin inonzi serotonergic agonist yakananga kune 5HT-2C receptor yakagamuchirwa kuti igare iine hutungamiri hwekufutisa kune varwere vane BMI ≥ 30 kg / m (2) kana BMI ≥ 27 kg / m (2) ine comorbidities ine chokuita nekufutisa.

Lorcaserin yakasarudzika yakasarudzika yakasarudzika serotonergic agonist yakagadzirirwa kuderedza njodzi dzinosangana nevamiriri vekare mukirasi ino. Pamishonga yekurapa, inotenderwa zvakanaka uye inogadzira kudzikira uremu zvine mwero asi zvine mutsindo nekunatsiridza kwakanyanya mu cardiometabolic paramita. Kubudirira kwekurapa kunofanirwa kuongororwa pamasvondo e12 (≥ 5% kurasikirwa uremu) kuona vanopindura vanozowana huwandu hwekuremerwa huremu uye kubatsirwa kwemetabolism kubva pakurapa kwenguva refu. Migumisiro yekuenderera mberi kwehutano hwemigumisiro yekuedza (CAMELLIA TIMI 61) ichasarudza basa re lorcaserin mukudzivirira kwekutanga kwechirwere cheshuga muvanhu vane uremu hwepamusoro / vakaoma uye kushandiswa kwayo muhuwandu hwehuwandu hwevarwere vane chirwere chemwoyo chakasimbiswa kana kuti multiple cardiovascular risk factors.

Kwatenga Lorcaserin hydrochloride Upfu?

Lorcaserin inoshandiswa kubatsira vanhu vakuru vane uremu kana kuti vane uremu uye vane matambudziko ehutano ane uremu kuti vaderedze uremu uye varambe vachiwana uremu ihwohwo. Lorcaserin inofanira kushandiswa pamwe chete nekuderedza calorie kudya uye chirongwa chekurovedza muviri. Lorcaserin iri mukirasi yemishonga inonzi serotonin receptor agonists. Inoshanda nekuwedzera manzwiro ekuzara kuitira kuti zvokudya zvishoma zvidyiwe.

Raw Lorcaserin hydrochloride Powder Testing Report-HNMR

Lorcaserin hydrochloride HNMR

Chii chinonzi HNMR uye HNMR spectrum inokuudza chii? H Nuclear Magnetic Resonance (NMR) spectroscopy inzira yekuongorora chemistry inoshandiswa mukudzora kwemhando uye tsvagiridzo yekuona zvirimo uye kuchena kwesample pamwe nemaitiro ayo mamorekuru. Semuyenzaniso, NMR inokwanisa kuongorora musanganiswa ane zvinozivikanwa makomboni. Kumakomisheni asingazivikanwe, NMR inogona kushandiswa kuenzanisa nekuona maraibhurari kana kufembera iyo yakakosha chimiro zvakananga. Kana iyo yekutanga dhizaini yazivikanwa, NMR inogona kushandiswa kuona mamolecular conformation mumhinduro pamwe nekudzidza zvimiro zvemuviri padanho remamorekuru senge conformational exchange, shanduko yechikamu, solubility, uye diffusion.

Lorcaserin hydrochloride (1431697-94-7) -COA

Lorcaserin hydrochloride (1431697-94-7) -COA

Nzira yekutenga Lorcaserin hydrochloride Upfu kubva kuAASraw?

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Reference

[1] Belviq (lorcaserin hydrochloride) piritsi [Eisai, Inc]”. DailyMed. Eisai, Inc. Nyamavhuvhu 2012. Yakachengetwa kubva kune yepakutanga musi wa21 Gumiguru 2013. Yakadzorerwa 21 Gumiguru 2013.

[2] "FDA inokumbira kubviswa kwemishonga inoderedza uremu Belviq, Belviq XR (lorcaserin) kubva pamusika". US Food and Drug Administration (FDA). 14 Ndira 2020. Yakadzorerwa 1 Kubvumbi 2020.

[3] "FDA Muchidimbu: FDA Inokumbira Kuzvidira Kubviswa Kwehuremu-Kurasikirwa Nemishonga Mushure meClinical Trial Inoratidza Kuwedzera Kuitika Kwekenza". FDA. 13 Kukadzi 2020.

[4] "Belviq XR (lorcaserin hydrochloride) mahwendefa akawedzerwa-kusunungurwa". US Food and Drug Administration (FDA). 26 Gumiguru 2016. Yakadzorerwa 14 Ndira 2020.

[5] "Drug Approval Package: Belviq (lorcaserin hydrochloride) Mahwendefa NDA #022529". US Food and Drug Administration (FDA). 7 Nyamavhuvhu 2012. Yakadzorerwa 14 Ndira 2020.


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